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托伐普坦中间体Tolvaptan1. 7-氯-1,2,3,4-四氢苯并[B]氮杂卓-5-酮 (CAS NO:160129-45-3)7-Chloro-1,2,3,4-tetrahydrobenzo[b] azepin-5-one2. 7-氯-1,2,3,4-四氢-1-(2-甲基-4-硝基苯甲酰基)-5H-1-苯并氮杂卓-5-酮7-Chloro-1,2,3,4-tetrahydro-1-(2-methyl-4-nitrobenzoyl)-5H-1-benzazepine-5-on (CAS NO:137982-91-3)3. 1-(4-氨基-2-甲基苯甲酰基)-7-氯-1,2,3,4-四氢-5H-1-苯并氮杂卓-5-酮1-(4-Amino-2-methylbenzoyl)-7-chloro-1,2,3,4-tetrahydro-5H-1-benzazepine-5-one(CAS NO:137977-97-0)4. N-[4-[(7-氯-2,3,4,5-四氢-5-氧代-1H-1-苯并氮杂卓-1-基)羰基]-3-甲基苯基]-2-甲基苯甲酰胺N-[4-[7-Chloro-2,3,4,5-tetrahydro-5-oxo-1H-1-benzazepine-1-yl)carbonyl]-3-methylphenyl]-2-methylbenzamide(CAS NO:137973-76-3)

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多佐胺中间体1. 多佐胺-2-13-(2-thienylthio)butyric acid  (CAS NO:133359-80-5)2. 多佐胺-2-2 5,6-dihydro 6- methyl-6H-thieno[2,3-b]thiopyran-2-sulfonamide-4-one3.  4,5-dihydro-6-methyl-6H-thieno[2,3-b] thiopyran-2-sulfonamide-4-ol 7,7,-dioxide 达泊西汀中间体1. (R)-(+)-3-氯-1-苯基-1-丙醇3-chloro-1-phenyl-propan-1-ol (CAS NO:100306-33-0)2. 3-(萘-4氧基)-1-苯基-1-丙醇3-(Naphthalen-4-yloxy)-1-Phenyl propan-1-ol3. 达泊西汀Dapoxetine (CAS NO:119356-77-3) 卡立普多中间体1. 5-甲基-5-丙基-1,3-二恶烷-2-酮 5-Methyl-5-Propyl-2-methyl Dioxanone (CAS NO:7148-50-7)2. 2-甲基-2-丙基-1,3-丙二醇异丙基氨基甲酸单酯N-Isopropyl-2-methyl-2-propyl-3-hydroxy propyl carbomate  (CAS NO:25462-17-3)

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卢帕他定中间体1.卢帕他定三盐酸盐(CAS NO:156611-76-6)2.卢帕他定(CAS NO:158876-82-5) 阿齐沙坦中间体1. 1-[(2'-(羟基脒基)[1,1-联苯基]-4-基)甲基]-2-乙氧基-1H-苯并咪唑-7-甲酸甲酯(CAS NO:147403-65-4)(Z)-Methyl 2-ethoxy-3-((2'-(N'-hydroxycarbaMiMidoyl)biphenyl-4-yl)Methyl)-3H-benzo[d] iMidazole-4-carboxylate2. 1-[(2'-[(乙氧羰基)氧基]脒基)[1,1-联苯基]-4-基)甲基]-2-乙氧基-1H-苯并咪唑-7-甲酸甲酯 1H-BenziMidazole-7-carboxylic acid, 1-[[2'-(2,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]Methyl] -2-ethoxy-, Methyl ester(CAS NO:147403-52-9)3. 阿齐沙坦 Azilsartan (CAS NO:147403-03-0)4. 4-(羟甲基)-5-甲基-[1,3]二氧杂环戊烯-2-酮4-(hidroximetil)-5-metil-1,3-dioxol-2-ona (CAS NO:91526-18-0)5. 阿齐沙坦酯 Azilsartan Medoxomil (CAS NO:863031-21-4) 

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鲁拉西酮中间体1. (1R,2R)-1,2-环己烷二甲醇 (1R,2R)-1,2-CYCLOHEXANEDIMETHANOL (CAS NO:65376-05-8)2. (R,R)-1,2-双(甲磺酰基氧基甲基)环己烷(R,R)-1,2-bis(methanesulfonyloxymethyl)cyclohexane (CAS NO:186204-35-3)3. (3AR,4S,7R,7AS) 4,7-亚甲基-1H-异吲哚-1,3(2H)-二酮(3aR,4S,7R,7aS) 4,7-Methano-1H-isoindole-1,3(2H)-dione (CAS NO:14805-29-9) 西咪匹韦中间体1. 反式-4-环己烯-1,2-二甲酸二乙酯DIETHYL TRANS-4-CYCLOHEXENE-1,2-DICARBOXYLATE (CAS NO:5048-50-0) 度鲁特韦中间体1.Methyl-5-(benzyloxy)-4-hydroxy-6-methylnicotinate  (CAS NO:906657-87-2)2.5-(benzyloxy)-4-hydroxy-6-(hydroxymethyl)nicotinic acid (CAS NO:906657-91-8)3.3-(benzyloxy)-5-(2,4-difluorobenzyl carbamoyl)4-hydroxy picolinic acid

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普鲁卡必利中间体1. 4-乙酰氨基-5-氯-2-羟基苯甲酸甲酯4-Acetylamino-5-Chloro-2-Hydroxybenzoic Acid Methyl Ester (CAS NO:24190-77-0)2. 4-氨基-5-氯-2,3-二氢苯并呋喃-7-羧酸4-Amino-5-chloro-2,3-dihydro-7-benzofurancarboxylic acid(CAS NO:123654-26-2)3. 1-(3-甲氧基丙基)-4-哌啶胺1-(3-Methoxypropyl)-4-piperidinamine (CAS NO:179474-79-4) 西尼必利中间体1. 4-AMino-2-ethoxy-5-nitrobenzoic Acid Methyl Ester (CAS NO:86718-17-4)2.西尼必利 CINITAPRIDE (CAS NO:66564-14-5) 

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加雷沙星中间体1.2-(Enzyl carbonyl)(1R)-5-bromo-2,3-dihydro-1-methyl-1H-isoindole (CAS NO:194805-13-5)2. (R)-5-bromo-1-methyl-2-tritylisoindoline (CAS NO:194805-14-6)3. Ethyl 7-bromo-1-cyclopropyl-8-(difluoromethoxy)-4-oxo-1,4-dihydroquinoline-3-carboxylate (CAS NO:194805-07-7)4.2-[(1R)-1-甲基-2-三苯甲基-2,3-二氢-1H-5-异吲哚基]硼酸二乙醇胺酯2,3-Dihydro-(1R)-methyl-5-(tetrahydro-4H-1,3,6,2-dioxazaborocin-2-yl)-2-(triphenylmethyl)-1H-isoindole(CAS NO:223595-20-8) 度洛西汀中间体1. S-(-)-N,N-二甲基-3-羟基-3-(2-噻吩)丙胺(S)-(-)-N,N-Dimethyl-3-hydroxy-3-(2-thienyl)propanamine (CAS NO:132335-44-5)2.3-甲基氨基-1-(2-噻吩基)-1-丙醇3-Methylamino-1-(2-thienyl)-1-propanol (CAS NO: 116539-55-0) 卢非酰胺中间体1. 1-[(2,6-二氟苯基)甲基]-1H-1,2,3-三唑-4-羧酸1-[(2,6-Difluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid  (CAS NO:166196-11-8)2. 4-氰基-1-(2,6-二氟苄基)-1H-1,2,3-三氮唑4-cyano-1-(2,6-difluorobenzyl)-1H-1,2,3-triazole (CAS NO:202003-06-3)

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尼卡地平中间体1. N-(2-氯乙基)-N-甲基苄胺盐酸盐benzyl-(2-chloroethyl)-methyl-azanium chloride CAS NO:23510-18-1 2. 2-(benzylmethylamino)ethyl acetoacetate (CAS NO:54527-65-0)3. 2-(3-硝基苯亚甲基)乙酰乙酸甲酯Methyl 3-nitrobenzylideneacetoacetate (CAS NO:39562-17-9)4. 4-(间硝基苯基)-2,6-二甲基-1,4-二氢-3,5-吡啶二羧酸二甲酯Dimethyl 4-(m-nitrophenyl)-2,6-dimethyl-1,4-dihydro-3,5-pyridinedicarboxylate (CAS NO:21881-77-6)5. 1,4-二氢-2,6-二甲基-4-(3-硝基苯基)吡啶-3,5-二甲酸单甲酯1,4-Dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic Acid 3-Methyl Ester (CAS NO:74936-72-4) 坦度螺酮中间体1.N-(4-bromobutyl)bicycle[2 2.1]heptane -2,3-di-exo –carboxamide (CAS NO:99095-09-7) 

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